Apabetalone
Supplier | MedChemExpress |
---|---|
Product # | HY-16652-25 mg |
CAS # | 1044870-39-4 |
Pricing | 25 mg, USD $240.0 |
Synonyms | RVX-208; RVX000222 |
MWt | 370.4 |
Formula | C₂₀H₂₂N₂O₅ |
Biological Activity | Apabetalone (RVX-208) is an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain. The IC50s are 87 μM and 0.51 μM for BD1 and BD2, respectively[1]. |
Purity | 99.86% |