LT052
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-130622-5 mg |
| CAS # | 2543545-44-2 |
| Pricing | 5 mg, USD $500.0 |
| Biological Activity | LT052 is a highly selective BET BD1 inhibitor with an IC50 of 87.7 nM. LT052 exhibits nanomolar BRD4 BD1 potency and 138-fold selectivity over BRD4 BD2 (IC50=12.130 μM). LT052 has anti-inflammatory activity and can be used for acute gout arthritis research[1]. |
| Purity | 98.49% |
| MWt | 449.48 |
| Formula | C₂₂H₁₉N₅O₄S |