CGP 78608 hydrochloride
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-107701 |
| CAS # | 1135278-54-4 |
| Pricing | inquire |
| Biological Activity | CGP 78608 hydrochloride is a highly potent and selective antagonist at the glycine-binding site of the NMDA receptor, with an IC50 of 6 nM. CGP 78608 acts as a potentiator of GluN1/GluN3A-mediated glycine currents, with an estimated EC50 in the low nM range (26.3 nM). Anticonvulsant activity[1][2]. |
| MWt | 414.58 |
| Formula | C₁₁H₁₄BrClN₃O₅P |