TPMPA
TPMPA is a selective and competitive GABAA-ρ antagonist with 8-fold selectivity for human recombinant ρ1 receptors over ρ2 receptors. TPMPA exhibits minimal effects on GABAA and GABAB receptors (Kb = 2.1 μM (antagonist), 320 μM (antagonist) and EC50 ~ 500 μM (weak agonist) for GABAA-ρ, GABAA and GABAB receptors, respectively).
Supplier | BOC Sciences |
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Product # | 182485-36-5 |
Pricing | Inquire |
Cas | 182485-36-5 |
Molecular Weight | 161.14 |
Molecular Formula | C6H12NO2P |
Canonical SMILES | CP(=O)(C1=CCNCC1)O |