TPMPA

TPMPA is a selective and competitive GABAA-ρ antagonist with 8-fold selectivity for human recombinant ρ1 receptors over ρ2 receptors. TPMPA exhibits minimal effects on GABAA and GABAB receptors (Kb = 2.1 μM (antagonist), 320 μM (antagonist) and EC50 ~ 500 μM (weak agonist) for GABAA-ρ, GABAA and GABAB receptors, respectively).
Supplier BOC Sciences
Product # 182485-36-5
Pricing Inquire
Cas 182485-36-5
Molecular Weight 161.14
Molecular Formula C6H12NO2P
Canonical SMILES CP(=O)(C1=CCNCC1)O
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