WDR5-IN-4

Supplier MedChemExpress
Product # HY-111753
CAS # 2407457-36-5
Pricing inquire
Biological Activity WDR5-IN-4 is an inhibitor of the WIN site of chromatin-associated WD repeat-containing protein 5 (WDR5), with a Kd of 0.1 nM. WDR5-IN-4 displaces WDR5 from chromatin and decreases the expression of associated genes, causing translational inhibition, nucleolar stress. Anti-cancer activity[1].
MWt 498.38
Formula C₂₅H₂₂Cl₂FN₅O

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