WDR5-IN-4
Supplier | MedChemExpress |
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Product # | HY-111753 |
CAS # | 2407457-36-5 |
Pricing | inquire |
Biological Activity | WDR5-IN-4 is an inhibitor of the WIN site of chromatin-associated WD repeat-containing protein 5 (WDR5), with a Kd of 0.1 nM. WDR5-IN-4 displaces WDR5 from chromatin and decreases the expression of associated genes, causing translational inhibition, nucleolar stress. Anti-cancer activity[1]. |
MWt | 498.38 |
Formula | C₂₅H₂₂Cl₂FN₅O |
Citations for this product:
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bioRxiv - Developmental Biology 2023Quote: ... WDR5-IN-4 (100 μg, MedChemExpress, HY-111753A), containing 0.05% Malachite Green reagent for tracing ...