R 59-022
Supplier | MedChemExpress |
---|---|
Product # | HY-107613-5 mg |
CAS # | 93076-89-2 |
Pricing | 5 mg, USD $350.0 |
Synonyms | DKGI-I; Diacylglycerol kinase inhibitor I |
MWt | 459.58 |
Formula | C₂₇H₂₆FN₃OS |
Biological Activity | R 59-022 (DKGI-I) is a diacylglycerol kinase inhibitor (IC50=2.8 μM). R 59-022 is a 5-HTR antagonist, and activates protein kinase C (PKC). R 59-022 potentiates thrombin-induced diacylglycerol production in platelets and inhibits phosphatidic acid production in neutrophils[1][2][3][4]. |
Purity | ≥99.0% |