FR 139317
FR 139317 is a selective Endothelin A receptor antagonist originated by Fujisawa. (Ki values are 1 nM and 7.3 μM at ETA and ETB subtypes respectively). No development was reported for the treatment of Cerebrovascular disorders, Coronary disorders, Diabetic nephropathies, Heart failure, Hypertension, Ischaemic heart disorders, Myocardial infarction and Renal failure.
| Supplier | BOC Sciences |
|---|---|
| Product # | 142375-60-8 |
| Pricing | Inquire |
| Cas | 142375-60-8 |
| Molecular Weight | 604.75 |
| Molecular Formula | C33H44N6O5 |
| Canonical SMILES | c12c(c(C[C@@H](NC([C@@H](NC(=O)N3CCCCCC3)CC(C)C)=O)C(=O)N[C@@H](C(O)=O)Cc3ncccc3)cn2C)cccc1 |