Eprenetapopt
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-19980-5 mg |
| CAS # | 5291-32-7 |
| Pricing | 5 mg, USD $84.0 |
| Synonyms | APR-246; PRIMA-1Met |
| MWt | 199.25 |
| Formula | C₁₀H₁₇NO₃ |
| Biological Activity | Eprenetapopt (APR-246) is a first-in-class, small molecule that restores wild-type p53 functions in TP53-mutant cells. Eprenetapopt triggers apoptosis in tumor cells. Eprenetapopt also targets the selenoprotein thioredoxin reductase 1 (TrxR1), a key regulator of cellular redox balance[1][2][3]. |
| Purity | ≥99.0% |