SB 271046 Hydrochloride
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-14336A-10 mM * 1 mL |
| CAS # | 209481-24-3 |
| Pricing | 10 mM * 1 mL, USD $152.0 |
| Synonyms | SB 271046A |
| MWt | 488.45 |
| Formula | C₂₀H₂₃Cl₂N₃O₃S₂ |
| Biological Activity | SB 271046 Hydrochloride (SB 271046A) is a potent, selective and orally active 5-HT6 receptor antagonist with pKi of 9.02, 8.55, and 8.81 for rat, pig and human, respectively. SB 271046 Hydrochloride is over 200 fold selective for the 5-HT6 receptor vs 55 other receptors, binding sites and ion channels. Anticonvulsant activity (EC50=0.16 μM)[1]. |
| Purity | 98.64% |