Pralsetinib
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-112301-5 mg |
| CAS # | 2097132-94-8 |
| Pricing | 5 mg, USD $130.0 |
| Synonyms | BLU-667 |
| MWt | 533.6 |
| Formula | C₂₇H₃₂FN₉O₂ |
| Biological Activity | Pralsetinib (BLU-667) is a highly potent, selective RET inhibitor. Pralsetinib (BLU-667) inhibits WT RET, RET mutants V804L, V804M, M918T and CCDC6-RET fusion with IC50s of 0.4, 0.3, 0.4, 0.4, and 0.4 nM, respectively[1]. |
| Purity | 99.56% |