GSK2801

Supplier MedChemExpress
Product # HY-15658-10 mM * 1 mL
CAS # 1619994-68-1
Pricing 10 mM * 1 mL, USD $88.0
Biological Activity GSK2801 is a potent, selective, orally active and cell active acetyl-lysine competitive BAZ2A and BAZ2B bromodomains inhibitor with Kd values of 136 nM and 257 nM, respectively. GSK2801 shows >50-fold selectivity for BAZ2A/B over BRD4[1].
MWt 371.45
Formula C₂₀H₂₁NO₄S
Feedback