GSK2801
Supplier | MedChemExpress |
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Product # | HY-15658-10 mM * 1 mL |
CAS # | 1619994-68-1 |
Pricing | 10 mM * 1 mL, USD $88.0 |
Biological Activity | GSK2801 is a potent, selective, orally active and cell active acetyl-lysine competitive BAZ2A and BAZ2B bromodomains inhibitor with Kd values of 136 nM and 257 nM, respectively. GSK2801 shows >50-fold selectivity for BAZ2A/B over BRD4[1]. |
MWt | 371.45 |
Formula | C₂₀H₂₁NO₄S |