Soraprazan
Supplier | MedChemExpress |
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Product # | HY-100414-1 mg |
CAS # | 261944-46-1 |
Pricing | 1 mg, USD $180.0 |
Synonyms | BYK61359 |
MWt | 367.44 |
Formula | C₂₁H₂₅N₃O₃ |
Biological Activity | Soraprazan (BYK61359) is a selective, reversible K-competitive inhibitor of the H,K-ATPase (Ki=6.4 nM), with an IC50 of 0.19 μM in gastric glands. Soraprazan binds to the H,K-ATPase with a Kd of 28.27 nM. Soraprazan shows immediate inhibition of acid secretion and is more than 2000-fold selective for H,K-ATPase over Na,K- and Ca-ATPases[1]. |
Purity | 99.69% |