TAK-828F
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-111509 |
| CAS # | 1854901-94-2 |
| Pricing | inquire |
| Biological Activity | TAK-828F is a potent, selective, and orally available retinoic acid receptor-related orphan receptor γt (RORγt) inverse agonist (binding IC50=1.9 nM, reporter gene IC50=6.1 nM). TAK-828F shows excellent RORγt isoforms selectivity (>5000-fold selectivity against human RORα and RORβ)[1]. |
| MWt | 509.57 |
| Formula | C₂₈H₃₂FN₃O₅ |