LY-288513
LY-288513 is a selective CCK2 receptor antagonist (IC50 values are 16 and > 30,000 nM for CCK2 and CCK1 respectively). LY-288513 displays anxiolytic and antipsychotic properties in vivo.
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD283 |
| CAS # | 147523-65-7 |
| Pricing | Customizable size, Inquiry |
| Synonym | LY-288513; LY 288513; LY288513. |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C22H18BrN3O2 |
| Exact Mass | 435.0582 |
| Molecular Weight | 436.31 |
| Elemental Analysis | C, 60.56; H, 4.16; Br, 18.31; N, 9.63; O, 7.33 |
| IUPAC/Chemical Name | 1-Pyrazolidinecarboxamide, N-(4-bromophenyl)-3-oxo-4,5-diphenyl-, (4S,5R)- |
| InChi Key | LMUQHXHWJWQXSD-PMACEKPBSA-N |
| InChi Code | InChI=1S/C22H18BrN3O2/c23-17-11-13-18(14-12-17)24-22(28)26-20(16-9-5-2-6-10-16)19(21(27)25-26)15-7-3-1-4-8-15/h1-14,19-20H,(H,24,28)(H,25,27)/t19-,20-/m0/s1 |
| SMILES Code | O=C(N1NC([C@@H](C2=CC=CC=C2)[C@@H]1C3=CC=CC=C3)=O)NC4=CC=C(Br)C=C4 |
| Appearance | Solid powder |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |