Flumazenil
Flumazenil is a specific benzodiazepine receptor antagonist primarily administered by injection. It is the only benzodiazepine receptor antagonist on the market today. Flumazenil is of benefit in patients who become excessively drowsy after benzodiazepines are used for either diagnostic or therapeutic procedures and it has been used as an antidote in the treatment of benzodiazepine overdoses.
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD473 |
| CAS # | 78755-81-4 |
| Pricing | Customizable size, Inquiry |
| Synonym | Flumazenil, Flumazepil, Anexate, Romazicon, Lanexat, Ro 15-1788, Ro 15 1788, Ro 151788 |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C15H14FN3O3 |
| Exact Mass | 303.1019 |
| Molecular Weight | 303.2884 |
| Elemental Analysis | C, 59.40; H, 4.65; F, 6.26; N, 13.85; O, 15.83 |
| IUPAC/Chemical Name | ethyl 8-fluoro-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate |
| InChi Key | OFBIFZUFASYYRE-UHFFFAOYSA-N |
| InChi Code | InChI=1S/C15H14FN3O3/c1-3-22-15(21)13-12-7-18(2)14(20)10-6-9(16)4-5-11(10)19(12)8-17-13/h4-6,8H,3,7H2,1-2H3 |
| SMILES Code | O=C(C1=C(CN2C)N(C=N1)C3=CC=C(F)C=C3C2=O)OCC |
| Appearance | White to off-white solid powder. |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO, not in water |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |
| Availability | 2 Weeks |