Palbociclib Isethionate
Palbociclib Isethionate is a highly selective inhibitor of CDK4/6 with IC50 of 11 nM/16 nM in cell-free assays. It shows no activity against CDK1/2/5, EGFR, FGFR, PDGFR, InsR, etc. Phase 3.
Supplier | Selleck Chemicals |
---|---|
Product # | S1579 |
Sku # | S1579-200mg |
Pricing | 200mg, $527.00 |
Citations for this product:
-
bioRxiv - Cell Biology 2020Quote: ... 2 μM Palbociclib Isethionate (CDK4i) (Cat. No. S1579, Selleck Chemicals), and 100 μM Ciprofloxacin (Cat ...
-
bioRxiv - Cancer Biology 2019Quote: ... Stocks of BRAF inhibitor PLX4720 (Catalog No. S1152) and CDK6 inhibitor palbociclib Isethionate (PD0332991, Catalog No. S1579) were purchased from Selleck Chemicals.