PF-3758309 hydrochloride
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-13007A |
| CAS # | 1279034-84-2 |
| Pricing | inquire |
| Biological Activity | PF-3758309 hydrochloride is a potent, orally available, and reversible ATP-competitive inhibitor of PAK4 (Kd= 2.7 nM; Ki=18.7 nM). PF-3758309 hydrochloride has the expected cellular functions of a PAK4 inhibitor: inhibition of anchorage-independent growth, induction of apoptosis, cytoskeletal remodeling, and inhibition of proliferation[1][2][3]. |
| MWt | 527.08 |
| Formula | C₂₅H₃₁ClN₈OS |