MT-802
MT-802 is a potent PROTAC that induces Bruton's tyrosine kinase (BTK) knockdown. MT-802 recruits BTK to the cereblon E3 ubiquitin ligase complex to trigger BTK ubiquitination and degradation via the proteasome. MT-802 has potential for treatment of C481S mutant chronic lymphocytic leukemia (CLL).
Supplier | Selleck Chemicals |
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Product # | S6966 |
Sku # | S6966-25mg |
Pricing | 25mg, $1797.00 |