Bifeprunox Mesylate
Bifeprunox, also known as DU-127090, is a partial dopamine and serotonin agonist potentially for the treatment of schizophrenia. Bifeprunox influences nicotine-seeking behaviour in response to drug-associated stimuli in rats. Bifeprunox suppresses in vivo VTA dopaminergic neuronal activity via D2 and not D3 dopamine autoreceptor activation.
| Supplier | Ace Therapeutics |
|---|---|
| Product # | SMD1440 |
| CAS # | 350992-13-1 (mesylate) |
| Pricing | Customizable size, Inquiry |
| Synonym | Bifeprunox; Bifeprunox Mesylate; DU-127090; DU 127090; DU127090. |
| Product Category | Lab-use Small Molecule Drugs |
| Chemical Formula | C25H27N3O5S |
| Molecular Weight | 481.567 |
| Elemental Analysis | C, 62.35; H, 5.65; N, 8.73; O, 16.61; S, 6.66 |
| IUPAC/Chemical Name | 7-(4-(Biphenyl-3-ylmethyl)piperazin-1-yl)benzoxazol-2(3H)-one methanesulfonate |
| InChi Key | ONWKHSGOYGLGPO-UHFFFAOYSA-N |
| InChi Code | InChI=1S/C24H23N3O2.CH4O3S/c28-24-25-21-10-5-11-22(23(21)29-24)27-14-12-26(13-15-27)17-18-6-4-9-20(16-18)19-7-2-1-3-8-19;1-5(2,3)4/h1-11,16H,12-15,17H2,(H,25,28);1H3,(H,2,3,4) |
| SMILES Code | O=C1OC2=C(N3CCN(CC4=CC(C5=CC=CC=C5)=CC=C4)CC3)C=CC=C2N1.CS(=O)(O)=O |
| Appearance | Solid powder |
| Purity | >98% (or refer to the Certificate of Analysis) |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| Storage Condition | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO |
| Shelf Life | >2 years if stored properly |
| Drug Formulation | This drug may be formulated in DMSO |
| Stock Solution Storage | 0 - 4℃ for short term (days to weeks), or -20℃ for long term (months). |
| HS Tariff Code | 2934.99.9001 |
| Availability | 2 Weeks |