Teglarinad chloride
Supplier | MedChemExpress |
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Product # | HY-10080-50 mg |
CAS # | 432037-57-5 |
Pricing | 50 mg, USD $2200.0 |
Synonyms | GMX1777; EB-1627 |
MWt | 672.6 |
Formula | C₃₀H₄₃Cl₂N₅O₈ |
Biological Activity | Teglarinad chloride (GMX1777) is a prodrug of GMX1778 (a nicotinamide phosphoribosyl transferase inhibitor). Teglarinad chloride exhibits antitumor activity in mice can be attributed to inhibition of NAMPT. Teglarinad chloride also enhances radiation efficacy, mediated by interference with DNA repair and antiangiogenesis[1][2]. |
Purity | 98.07% |