Bimiralisib

Supplier MedChemExpress
Product # HY-12868-10 mg
CAS # 1225037-39-7
Pricing 10 mg, USD $140.0
Synonyms PQR309
MWt 411.38
Formula C₁₇H₂₀F₃N₇O₂
Biological Activity Bimiralisib (PQR309) is a potent, brain-penetrant, orally bioavailable, pan-class I PI3K/mTOR inhibitor with IC50s of 33 nM, 451 nM, 661 nM, 708 nM and 89 nM for PI3Kα, PI3Kδ, PI3Kβ, PI3Kγ and mTOR, respectively. Bimiralisib is an mTORC1 and mTORC2 inhibitor.
Purity 98.74%
Feedback