Varenicline
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-10019-5 mg |
| CAS # | 249296-44-4 |
| Pricing | 5 mg, USD $84.0 |
| Synonyms | CP 526555 |
| MWt | 211.26 |
| Formula | C₁₃H₁₃N₃ |
| Biological Activity | Varenicline (CP 526555) is a potent partial agonist for α4β2 nicotinic acetylcholine receptor (nAChR) with an EC50 value of 2.3 μM. Varenicline is a full agonist for α3β4 and α7 nAChRs with EC50 values of 55 μM and 18 μM, respectively[1]. Varenicline is a nicotinic ligand based on the structure of cytisine, has the potential for smoking cessation treatment[2]. |
| Purity | 99.70% |