GI-530159
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-W013712-100 mg |
| CAS # | 69563-88-8 |
| Pricing | 100 mg, USD $50.0 |
| Biological Activity | GI-530159 is a selective, mechanosensitive opener of TREK1 (K2P2.1) and TREK2 (K2P10.1) channels, with an EC50 of 0.76 μM for TREK1. GI-530159 displays selectivity for TREK1/2 over TRAAK, TASK3 and other potassium channels. GI-530159 reduces rat dorsal root ganglion neuron excitability[1]. |
| Purity | ≥98.0% |
| MWt | 518.45 |
| Formula | C₂₇H₂₀F₆N₂O₂ |