RPR-260243
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-16915-5 mg |
| CAS # | 668463-35-2 |
| Pricing | 5 mg, USD $264.0 |
| Biological Activity | RPR-260243, a potent activator of human ether-a-go-go-related gene (hERG), slows deactivation and attenuates inactivation of hERG1 channels. RPR260243-modified HERG currents are inhibited by Dofetilide (IC50=58 nM). RPR260243 displays no activator-like effects on other voltage-dependent ion channels, including the closely related ERG3 K+ channel[1][2]. |
| Purity | 99.37% |
| MWt | 510.5 |
| Formula | C₂₈H₂₅F₃N₂O₄ |