RBN012759
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-136979-10 mM * 1 mL |
| CAS # | 2360851-29-0 |
| Pricing | 10 mM * 1 mL, USD $440.0 |
| Biological Activity | RBN012759 is a potent, selective and orally active inhibitor of PARP14, with an IC50 of <3 nM. RBN012759 displays 300-fold selectivity over the monoPARPs and 1000-fold selectivity over the polyPARPs. RBN012759 decreases pro-tumor macrophage function and elicits inflammatory responses in tumor explants[1]. |
| Purity | 99.88% |
| MWt | 378.46 |
| Formula | C₁₉H₂₃FN₂O₃S |