Belzutifan
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-125840-10 mM * 1 mL |
| CAS # | 1672668-24-4 |
| Pricing | 10 mM * 1 mL, USD $826.0 |
| Synonyms | PT2977; MK-6482 |
| MWt | 383.34 |
| Formula | C₁₇H₁₂F₃NO₄S |
| Biological Activity | Belzutifan (PT2977) is an orally active and selective HIF-2α inhibitor with an IC50 of 9 nM. Belzutifan, as a second-generation HIF-2α inhibitor, increases potency and improves pharmacokinetic profile. Belzutifan is a potential treatment for clear cell renal cell carcinoma (ccRCC)[1]. |
| Purity | 99.73% |