ESI-05
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-117656-5 mg |
| CAS # | 5184-64-5 |
| Pricing | 5 mg, USD $60.0 |
| Synonyms | NSC 116966 |
| MWt | 274.38 |
| Formula | C₁₆H₁₈O₂S |
| Biological Activity | ESI-05 (NSC 116966) is a specific antagonist of EPAC2 (exchange protein directly activated by cAMP 2), with an IC50 of 0.4 µM. ESI-05 (NSC 116966) inhibits cAMP-mediated activation of EPAC2 as well as EAPC2 mediated Rap1 activation[1]. |
| Purity | 99.94% |