RQ-00203078

Supplier MedChemExpress
Product # HY-18662-100 mg
CAS # 1254205-52-1
Pricing 100 mg, USD $450.0
Biological Activity RQ-00203078 is a highly selective, potent and orally active TRPM8 antagonist with IC50s of 5.3 nM and 8.3 nM for rat and human TRPM8 channels, respectively. RQ-00203078 shows little inhibitory action against TRPV1, TRPA1, TRPV4, or TRPM2 channels[1][2].
Purity 99.84%
MWt 554.85
Formula C₂₁H₁₃ClF₆N₂O₅S
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