RQ-00203078
Supplier | MedChemExpress |
---|---|
Product # | HY-18662-100 mg |
CAS # | 1254205-52-1 |
Pricing | 100 mg, USD $450.0 |
Biological Activity | RQ-00203078 is a highly selective, potent and orally active TRPM8 antagonist with IC50s of 5.3 nM and 8.3 nM for rat and human TRPM8 channels, respectively. RQ-00203078 shows little inhibitory action against TRPV1, TRPA1, TRPV4, or TRPM2 channels[1][2]. |
Purity | 99.84% |
MWt | 554.85 |
Formula | C₂₁H₁₃ClF₆N₂O₅S |