BX795
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-10514-200 mg |
| CAS # | 702675-74-9 |
| Pricing | 200 mg, USD $1080.0 |
| Biological Activity | BX795 is a potent and selective inhibitor of PDK1, with an IC50 of 6 nM. BX795 is also a potent and relatively specific inhibitor of TBK1 and IKKɛ, with an IC50 of 6 and 41 nM, respectively. BX795 blocks phosphorylation of S6K1, Akt, PKCδ, and GSK3β, and has lower selectivity over PKA, PKC, c-Kit, GSK3β etc. BX795 modulates autophagy[1][2][3][4]. |
| Purity | 99.06% |
| MWt | 591.47 |
| Formula | C₂₃H₂₆IN₇O₂S |