Umbralisib
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-12279-10 mg |
| CAS # | 1532533-67-7 |
| Pricing | 10 mg, USD $220.0 |
| Synonyms | TGR-1202; RP5264 |
| MWt | 571.55 |
| Formula | C₃₁H₂₄F₃N₅O₃ |
| Biological Activity | Umbralisib (TGR-1202) is a novel PI3Kδ inhibitor, with IC50 and EC50 of 22.2 nM and 24.3 nM, respectively; Umbralisib (TGR-1202) is also active against CK1ε, with an EC50 value of 6.0 μM. |
| Purity | ≥98.0% |