E7449

Supplier MedChemExpress
Product # HY-12418-50 mg
CAS # 1140964-99-3
Pricing 50 mg, USD $900.0
Biological Activity E7449 is a potent PARP1 and PARP2 inhibitor and also inhibits TNKS1 and TNKS2, with IC50s of 2.0, 1.0, ∼50 and ∼50 nM for PARP1, PARP2, TNKS1 and TNKS2, respectively, using 32P-NAD+ as substrate.
Purity ≥98.0%
MWt 317.34
Formula C₁₈H₁₅N₅O
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