MS1943
| Supplier | MedChemExpress |
|---|---|
| Product # | HY-133129-10 mg |
| CAS # | 2225938-17-8 |
| Pricing | 10 mg, USD $1300.0 |
| Biological Activity | MS1943 is a first-in-class, orally bioavailable EZH2 selective degrader, with an IC50 of 120 nM. MS1943 significantly reduces EZH2 protein levels in numerous triple-negative breast cancer (TNBC) and other cancer and noncancerous cell lines. MS1943 effectively blocks proliferation of multiple TNBC and other cancer cell lines[1]. |
| Purity | 98.18% |
| MWt | 718.93 |
| Formula | C₄₂H₅₄N₈O₃ |